Coluracetam ugu fiican (135463-81-9) Soo-saare - Cofttek

Coluracetam (135463-81-9)

Waxaa laga yaabaa 8, 2021

Cofttek waa soo saaraha budada Coluracetam ee ugu fiican Shiinaha. Warshadeena waxay leedahay nidaam maareyn wax soo saar oo dhameystiran (ISO9001 & ISO14001), oo leh awood wax soo saar bille ah 160kg.

 


Status: In Mass Production
Unugga: 1kg / bac, 25kg / Drum

Coluracetam (135463-81-9) Smamnuucista

Name: Coluracetam
CAS: 135463-81-9
xagiisayna 98%
Qaaciddada Molecular: C19H23N3O3
Miisaanka kelli: 341.411 g / moll
Dhibcaha Biyaha: N / A
Magaca kiimikada: N-(2,3-dimethyl-5,6,7,8-tetrahydrofuro[2,3-b]quinolin-4-yl)-2-(2-oxopyrrolidin-1-yl)acetamide

MKC-231

bci-540

micne ah: Coluracetam; BCI-540; MKC-231; BCI 540; MKC 231; BCI540; MKC231.
Furaha gudaha: PSPGQHXMUKWNDI-UHFFFAOYSA-N
Kala badh: N / A
Xalka: Dajinta DMSO
Xaaladda Kaydinta: Qalalan, madow iyo 0 - 4 C muddo gaaban (maalmo illaa toddobaadyo) ama -20 C muddo dheer (bilo illaa sannado)
Codsiga: qaydhiin Budada Coluracetam (MKC-231) is a synthetic racetam drug purported to be a nootropic compound.
Imaanshaha: budada crystalline cad

 

Coluracetam (135463-81-9) NMR Spectrum

Coluracetam (135463-81-9) NMR Spectrum

Haddii aad u baahan tahay COA, MSDS, HNMR qayb kasta oo badeecad ah iyo macluumaad kale ah, fadlan la soo xiriir annaga maareeyaha suuq gaynta.

 

waa maxay Coluracetam (135463-81-9)?

Root Coluracetam budada (MKC-231) waa daroogada jilicsan ee loo yaqaan 'synthetic drug prodetam' oo loo yaqaan 'nootropic compound'. Ma hayo jiritaan balaaran oo cadeyn ah, laakiin farsamooyinka ficilka (iyo sidoo kale qaabdhismeed) waxay u muuqdaan inay aad u kala duwan yihiin xeryahooda kale sida Piracetam ama Aniracetam.

Raw Coluracetam powder appears to interact with a process known as high affinity choline uptake (HACU for short), which is the rate-limiting step of drawing choline into a neuron for synthesis into the neurotransmitter acetylcholine. Increasing the HACU rate appears to increase the activity of cholinergic neurons, so it is a desired target for kobcinta garashada.

 

Coluracetam (135463-81-9) faa'iidooyinka

  • Hagaajinta Xusuusta iyo Barashada
  • Hagaajinta Akhriska Akhriska iyo Soo-Celinta Bilaashka ah
  • Hagaajinta Garashada Waqtiga-Dheer
  • Yareeyaan Murugada-Niyad jabka
  • Kordhinta suurtogalka ah ee Neurogenesis
  • Hagaajin kartaa Naafonimada Maskaxda
  • Hagaajinta Aragga
  • Calaamadaha loo yaqaan 'Irritable Bowel Syndrome Syndrome' oo la hagaajiyo
  • Isticmaalka madadaalada ee Coluracetam

 

Coluracetam (135463-81-9) isticmaalka

Coluracetam (INN) (code name BCI-540; formerly MKC-231) powder is a nootropic agent of the racetam family. Waxaa markii hore soo saaray oo tijaabisay Shirkadda Mitsubishi Tanabe Pharma ee cudurka Alzheimers. Ka dib markii daawadu ay ku guul darreysatay inay gaarto dhammaadka tijaabooyinkeeda caafimaad, waxaa shati u siisay BrainCells Inc si loo baaro xanuunka weyn ee niyad-jabka (MDD), kaas oo ka horreeyay in lagu abaalmariyo deeqda "Barnaamijka Daahfurka Daawaynta u Qalma" ee gobolka California.

 

Coluracetam (135463-81-9) qiyaasta

Cilmi-baarista ugu badan ee coluracetam waxaa lagu sameeyaa xayawaanka halkii aadanuhu, sidaa daraadeed ma jiraan tilmaamo daweyn oo guud ahaan loo aqbalo. Qiyaasta qiyaasta firfircoon ee guud ayaa guud ahaan lagu qeexaa sida xmUMX-5 mg. Isticmaalayaasha coluracetam ayaa soo sheegay in qiyaaso kala duwan oo qiyaas ah loo maamulo labadaba afka iyo lakulanka.

Jawaab celinta isticmaalaha ayaa sidoo kale sheegtay in dulqaadashada budada coluracetam ay si dhakhso leh u horumarin karto. Sida dawooyinka oo dhan, gaar ahaan nootropics, waxaa fiican inaad ku bilowdo qadar yar iyo inaad si tartiib tartiib ah kor ugu qaadatid qiyaasta sida jidhkaagu u falcelinayo una qaabeeyo daawada. Coluracetam waa mid aan sun ahayn waxaana loo tixgeliyaa inuu yahay mid dulqaad badan oo badbaado leh.

 

Budada Coluracetam for sale(Xagee laga iibsadaa budada Coluracetam ee badan)

Shirkadeena waxay ku raaxaysataa cilaaqaadka muddada dheer macaamiisheena sababtoo ah waxaan diirada saarnaa macaamiisha adeegga iyo bixinta alaabta weyn. Haddii aad xiisaynayso badeecadeena, waxaan la jaanqaadi karnaa qaabeynta amarrada si aan ugu haboono baahidaada gaarka ah iyo waqtigeenna degdegga ah ee amarrada oo damaanad qaadaya inaad badeecaddeena si weyn u dhadhamin doonto waqtiga. Waxaan sidoo kale diirada saarnaa adeegyada qiimaha lagu daray. Waxaan diyaar u nahay su'aalaha adeegga iyo macluumaadka aan ku taageerno ganacsigaaga.

We are an professional Coluracetam powder supplier for several years, we supply alaabooyin leh tartan qiimaha, iyo badeecadayadu waa tayada ugu sareysa waxaana lagu sameeyaa baaritaan adag, madax-bannaan si loo hubiyo inay ammaan u tahay isticmaalka adduunka oo dhan.

 

tixraacyada

[1] Akaike A, iyo al. (1998). Saamaynta badbaadada ee MKC-231, oo ah kobciyaha sare ee kor u qaadista xayeysiinta, ee ku saabsan 'glutamate cytotoxicity' ee neur-mareenka dhaqanka. Jpn J Farmasiil.

[2] Bessho, T., Takashina, K., Tabata, R., Ohshima, C., Chaki, H., Yamabe, H., Egawa, M., Tobe, A., & Saito, K. (1996). Saameynta nuxurka sare ee kor u qaadista koritaanka kor u qaadista 2- (2-oxopyrrolidin-1-yl) -N- (2,3-dimethyl-5,6,7,8-tetrahydrofuro [2,3-b] quinolin-4- yl) acetoamide oo ku saabsan cilladaha barashada suuxdinta biyaha ee jiirka. Arzneimittel-Forschung, 46 (4), 369-373.

[3] Murai, S., Saito, H., Abe, E., Masuda, Y., Odashima, J., & Itoh, T. (1994). MKC-231, kor u qaadista qashinka, waxay hagaajineysaa hoos u dhaca xusuusta iyo hoos u dhaca hippocampal acetylcholine oo ay sababtay ethylcholine aziridinium ion ee jiirka. Joornaalka Gudbinta Neural, 98 (1), 1-13. Doi: 10.1007 / bf01277590.

[4] Takashina K, Bessho T, Mori R, Eguchi J, Saito K. MKC-231, kor u qaadista kororka ee choline: (2) Saamaynta isugeynta iyo siideynta acetylcholine ee jiirka AF64A-daweynta. J Neural Transm (Vienna). 2008 Jul; 115 (7): 1027-35. doi: 10.1007 / s00702-008-0048-1. PubMed PMID: 18446264.

[5] Shirayama Y, Yamamoto A, Nishimura T, Katayama S, Kawahara R. Soo-jeedinta ku xigta ee kor u qaadista choline-ka MKC-231 waxay ka hortageysaa yaraanta dabeecadda dabeecadda-yaraanta dabeecadda iyo yaraynta septal cholinergic neurons ee jiirka. Eur Neuropsychopharmacol. 2007 Sep; 17 (9): 616-26. PubMed PMID: 17467960.

 


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